SCHEMBL25366451

SCHEMBL25366451

Fc1cccc(CC2CNC(=S)N2)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.40
MAPK1 P28482 1/20 0.40
PLG P00747 1/20 0.39
DBH P09172 1/20 0.38
P2RX7 Q99572 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
MIF P14174 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30528718 1.00 NPC1 (0.41) NPC1HTTMAPK1PLGDBH
SCHEMBL30528574 0.82 POLB (0.39) TAAR1MEN1ALDH1A1KMT2A
SCHEMBL25365104 0.82 KMT2A (0.42) HTTDBHTAAR1ALDH1A1KMT2A
SCHEMBL25367612 0.82 POLB (0.39) TAAR1MEN1ALDH1A1KMT2A
SCHEMBL30528591 0.82 KMT2A (0.42) HTTDBHTAAR1ALDH1A1KMT2A
SCHEMBL25365107 0.82 KMT2A (0.42) HTTDBHTAAR1ALDH1A1KMT2A
SCHEMBL25365743 0.81 ALDH1A1 (0.36) PLGDBHMEN1ALDH1A1KMT2A
SCHEMBL1598073 0.80 MEN1 (0.47) MEN1ALDH1A1KMT2A
SCHEMBL25366852 0.71 SMN1; SMN2 (0.36) HTTMAPK1MEN1ALDH1A1KMT2A
SCHEMBL25367156 0.71 MEN1 (0.37) DBHMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240018125-A1 CYCLIC ISOTHIOUREA DERIVATIVES AS CXCR4 MODULATORS ERMIUM THERAPEUTICS (FR) 2024-01-18 US disclosed
EP-4217353-A1 CYCLIC ISOTHIOUREA DERIVATIVES AS CXCR4 MODULATORS Ermium Therapeutics (FR) 2023-08-02 EP disclosed
WO-2022064075-A1 CYCLIC ISOTHIOUREA DERIVATIVES AS CXCR4 MODULATORS ERMIUM THERAPEUTICS (FR) 2022-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240018125-A1 CYCLIC ISOTHIOUREA DERIVATIVES AS CXCR4 MODULATORS CXCR4, CXCR1, CXCL12 NPC1 2463/4885HTT 4663/4885MAPK1 1156/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.