Pyrimidine

Pyrimidine

SCHEMBL25385683

NC=C(C(N)=O)c1ccccc1.c1cncnc1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
SARM1 Q6SZW1 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
SIRT4 Q9Y6E7 1/20 0.42
CYP2C19 P33261 4/20 0.41
CYP3A4 P08684 4/20 0.41
POLB P06746 2/20 0.41
PARP1 P09874 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17397067 0.87 TDP1 (0.52) KMT2AMEN1F7F3CYP2C19
Hydrochloric Acid SCHEMBL28280655 0.85 CYP2C19 (0.50) KMT2AMEN1F7F3CYP2C19
Acetic Acid SCHEMBL28542071 0.82 TSHR (0.46) KMT2AMEN1CYP2C19CYP3A4POLB
SCHEMBL15758917 0.81 F7 (0.61) F7F3SARM1SIRT2SIRT6
Benzamide SCHEMBL27841146 0.77 CYP3A4 (0.70) KMT2AMEN1NPC1RAB9AF7
SCHEMBL21074576 0.74 MKNK1 (0.67) NPC1RAB9AF7F3SARM1
SCHEMBL21074472 0.74 MKNK1 (0.67) NPC1RAB9AF7F3SARM1
Benzoic Acid SCHEMBL3313836 0.73 NAPRT (0.67) KMT2AMEN1CYP2C19CYP3A4TSHR
Benzophenone SCHEMBL4016306 0.73 KMT2A (0.71) KMT2AMEN1NPC1RAB9ACYP2C19
SCHEMBL7118621 0.73 AKR1C1 (0.59) KMT2AMEN1CYP2C19CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3658552-B1 PROCESS FOR PREPARING N-(5-((4-(4-((DIMETHYLAMINO)METHYL)-3-PHENYL-1H-PYRAZOL-1-YL)PYRIMIDIN-2-YL)AMINO)-4-METHOXY-2-MORPHOLINOPHENYL)ACRYLAMIDE BY REACTING THE CORRESPONDING AMINE WITH A 3-HALO-PROPIONYL CHLORIDE YUHAN CORP (KR) 2023-09-13 EP disclosed
CN-104788427-A 3-(2-pyrimidine amino) phenyl acrylic amide compound and application thereof PHARMARESOURCES SHANGHAI CO LTD 2015-07-22 CN disclosed
CN-104788427-A 3-(2-pyrimidine amino) phenyl acrylic amide compound and application thereof PHARMARESOURCES SHANGHAI CO LTD 2015-07-22 CN disclosed