SCHEMBL25404197

SCHEMBL25404197

Nc1ncc2c(I)c[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 12/20 0.42
CDK5 Q00535 10/20 0.42
CDK5R1 Q15078 10/20 0.42
MAPK1 P28482 1/20 0.41
CHEK1 O14757 1/20 0.38
ALDH1A1 P00352 1/20 0.36
CCNT1 O60563 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
CCNA1 P78396 2/20 0.36
PDPK1 O15530 1/20 0.34
BRD4 O60885 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAP3K11 Q16584 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25158173 0.78 AXL (0.48) CLK1CDK5CDK5R1MAPK1ALDH1A1
SCHEMBL17769864 0.77 MAP3K14 (0.38) CLK1CDK5CDK5R1ALDH1A1CCNT1
SCHEMBL12120921 0.77 TYRO3 (0.42) MAPK1CHEK1BRD4
SCHEMBL30475606 0.77 TYRO3 (0.42) MAPK1CHEK1BRD4
SCHEMBL13219255 0.73 MAPK1 (0.38) CLK1CDK5CDK5R1MAPK1CHEK1
SCHEMBL25401085 0.73 CHUK (0.51)
SCHEMBL311676 0.72 RPS6KA5 (0.45) CLK1CDK5MAPK1CHEK1CDK2
SCHEMBL23451864 0.72 CDK2 (0.53) CLK1CDK5CCNT1CCNA2CDK2
SCHEMBL4697304 0.69 RET (0.41) ALDH1A1CDK2PDPK1CYP3A4
SCHEMBL30822335 0.69 RET (0.41) ALDH1A1CDK2PDPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023177351-A1 NF ҚB INDUCING KINASE INHIBITORS AND METHODS THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-09-21 WO disclosed