SCHEMBL2540686

SCHEMBL2540686

COc1cc(-c2ccc3[nH]c(=O)n(CC4CC4)c3c2)cc(OC)c1OC

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 11/20 0.58
GRIN2B Q13224 11/20 0.58
MAP3K11 Q16584 4/20 0.53
PGR P06401 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
TP53 P04637 1/20 0.41
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL723941 0.80 GRIN1 (0.73) GRIN1GRIN2BMAP3K11
SCHEMBL29888611 0.73 GRIN1 (1.00) GRIN1GRIN2BMAP3K11
SCHEMBL20134253 0.73 GRIN1 (1.00) GRIN1GRIN2BMAP3K11
SCHEMBL11893902 0.73 GRIN1 (0.51) GRIN1GRIN2BL3MBTL1
SCHEMBL11893965 0.73 GRIN1 (0.51) GRIN1GRIN2BL3MBTL1
SCHEMBL20357946 0.72 MAPK9 (0.54) GRIN1GRIN2B
SCHEMBL11893888 0.71 GRIN1 (0.52) GRIN1GRIN2BL3MBTL1
SCHEMBL11893887 0.71 GRIN1 (0.52) GRIN1GRIN2BL3MBTL1
SCHEMBL11221627 0.70 PLD2 (0.43) GRIN1GRIN2BHTR7
SCHEMBL20134376 0.70 GRIN1 (1.00) GRIN1GRIN2BMAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed