SCHEMBL254123

SCHEMBL254123

COc1cc(/C=C/C(=O)N2CCC=CC2=O)cc(O)c1OCCN

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.71
TP53 P04637 3/20 0.71
MAPT P10636 3/20 0.71
SMN1; SMN2 Q16637 2/20 0.71
HSD17B10 Q99714 2/20 0.71
LMNA P02545 2/20 0.71
STAT3 P40763 2/20 0.71
CYP1A2 P05177 1/20 0.71
HIF1A Q16665 1/20 0.71
PSMB11 A5LHX3 1/20 0.71
PSMA7 O14818 1/20 0.71
NPC1 O15118 1/20 0.71
FOXO3 O43524 1/20 0.71
MITF O75030 1/20 0.71
CYP3A4 P08684 1/20 0.71
PSMB1 P20618 1/20 0.71
PSMA1 P25786 1/20 0.71
PSMA2 P25787 1/20 0.71
PSMA3 P25788 1/20 0.71
PSMA4 P25789 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173087 0.95 ALDH1A1 (0.78) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL98548 0.91 ALDH1A1 (0.71) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL19295194 0.86 ALDH1A1 (0.80) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL15444232 0.84 ALDH1A1 (0.77) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL173090 0.84 ALDH1A1 (0.83) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
Piplartine SCHEMBL2465593 0.84 ALDH1A1 (1.00) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
Piplartine SCHEMBL173092 0.84 ALDH1A1 (1.00) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
(Z)-Piplartine SCHEMBL30013548 0.84 ALDH1A1 (1.00) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL173089 0.83 ALDH1A1 (0.75) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10
SCHEMBL15444220 0.83 ALDH1A1 (0.75) ALDH1A1TP53MAPTSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030408-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CANCER CANTHERA THERAPEUTICS, INC. (US) 2012-03-08 WO disclosed