SCHEMBL25415263

SCHEMBL25415263

[O-][n+]1ccc(C(F)(F)F)cc1C(F)F

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331680 0.72 KIF11 (0.34) TSHRMAPK1S1PR1
SCHEMBL2145857 0.72 PDE2A (0.34) TSHRMAPK1S1PR1
SCHEMBL7412520 0.69 TSHR (0.31) TSHRMAPK1S1PR1
SCHEMBL17816206 0.69 KIF11 (0.37) TSHRMAPK1S1PR1
SCHEMBL19191095 0.68 TACR1 (0.34) TSHRMAPK1
SCHEMBL2331693 0.67 DRD4 (0.40)
SCHEMBL2334903 0.65 S1PR1 (0.53) TSHRS1PR1
SCHEMBL11818712 0.64 PTPN5 (0.35) TSHRMAPK1S1PR1
SCHEMBL4901404 0.63 KIF11 (0.45)
SCHEMBL16505901 0.63 CFTR (0.49) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023169573-A1 POLθ INHIBITOR 武汉人福创新药物研发中心有限公司 2023-09-14 WO disclosed
CN-116730979-A Pol theta inhibitor 武汉人福创新药物研发中心有限公司 2023-09-12 CN disclosed