SCHEMBL2543211

SCHEMBL2543211

COc1ccc2nccc(CC(=O)[C@H]3CC[C@H](NC(=O)OCc4ccccc4)CC3)c2n1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
GAA P10253 1/20 0.52
TSHR P16473 1/20 0.50
KCNH2 Q12809 5/20 0.43
DPP4 P27487 3/20 0.41
DPP7 Q9UHL4 3/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
ACHE P22303 2/20 0.41
EPHX1 P07099 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2543208 1.00 ALDH1A1 (0.52) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2541639 0.85 ALDH1A1 (0.45) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2541635 0.85 ALDH1A1 (0.45) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2543399 0.85 DPP4 (0.47) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2535504 0.85 DPP4 (0.47) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2535506 0.85 DPP4 (0.47) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2543394 0.85 DPP4 (0.47) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2538301 0.82 ALDH1A1 (0.41) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL2538299 0.82 ALDH1A1 (0.41) ALDH1A1GAATSHRKCNH2DPP4
SCHEMBL1223261 0.81 ALDH1A1 (0.45) ALDH1A1GAATSHRKCNH2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094267-B1 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2015-04-22 EP disclosed
US-8044044-B2 4-(1-amino-ethyl)-cyclohexylamine derivatives ACTELION PHARMACEUTICAL LTD. (CH) 2011-10-25 US disclosed
EP-2094267-A2 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-09-02 EP disclosed
WO-2008078305-A2 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-03 WO disclosed