SCHEMBL25463299

SCHEMBL25463299

CCc1c(C)ncnc1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
HTT P42858 2/20 0.32
GALR3 O60755 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
PDE10A Q9Y233 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.31
MAPT P10636 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
KDM5A P29375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16591438 0.87 PDPK1 (0.41) PDPK1HSD17B10LMNASMN1; SMN2CYP1A2
SCHEMBL29450983 0.82 PDPK1 (0.35) PDPK1HSD17B10LMNASMN1; SMN2MAPT
SCHEMBL22139947 0.82 PDPK1 (0.35) PDPK1HSD17B10LMNASMN1; SMN2MAPT
SCHEMBL22139943 0.82 HSD17B10 (0.38) PDPK1HSD17B10LMNATSHRKDM4E
SCHEMBL25517393 0.81 TSHR (0.44) LMNASMN1; SMN2HTTCYP1A2CYP2C9
SCHEMBL463190 0.79 CDC7 (0.39) NOS3NOS2ALDH1A1MEN1KMT2A
SCHEMBL13535769 0.77 HSD17B10 (0.33) PDPK1HSD17B10KDM4EKMT2A
SCHEMBL25734277 0.74 MEN1 (0.32) PDPK1HSD17B10MAPK1ALDH1A1MEN1
SCHEMBL13848218 0.74 NOS3 (0.32) CYP1A2CYP2D6CYP2C9CYP2C19NOS3
SCHEMBL12051534 0.73 PDPK1 (0.41) PDPK1HSD17B10LMNASMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023083297-A1 SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2023-05-19 WO disclosed
WO-2023083286-A1 SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2023-05-19 WO disclosed