SCHEMBL25473160

SCHEMBL25473160

C/C(=N\C=O)c1ccc(-c2scnc2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
VHL P40337 8/20 0.49
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
KDM4E B2RXH2 2/20 0.33
PKM P14618 1/20 0.33
ELOC Q15369 2/20 0.32
ELOB Q15370 2/20 0.32
P2RX3 P56373 1/20 0.32
P2RX2 Q9UBL9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23880997 0.79 VHL (0.60) VHLPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL24880893 0.75 VHL (0.52) VHLPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28610139 0.74 VHL (0.55) VHLKDM4EPKM
SCHEMBL26384247 0.73 VHL (0.50) VHLKDM4EPKMELOCELOB
Hydrochloric Acid SCHEMBL28668471 0.73 VHL (0.54) VHLKDM4EPKM
SCHEMBL19600685 0.71 VHL (0.54) VHLKDM4EPKMELOCELOB
SCHEMBL24440459 0.71 VHL (0.51) VHLKDM4EPKMELOCELOB
SCHEMBL23037352 0.71 VHL (0.51) VHLKDM4EPKMELOCELOB
SCHEMBL24327249 0.71 VHL (0.55) VHLKDM4EELOCELOB
SCHEMBL19661678 0.70 VHL (0.53) VHLKDM4EPKMELOCELOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081759-A1 BIFUNCTIONAL PI3K-ALPHA INHIBITORS AND USES THEREOF RELAY THERAPEUTICS, INC. (US) 2023-05-11 WO disclosed