SCHEMBL25474175

SCHEMBL25474175

CC[C@H]1C[C@H](N)CCN1C

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GNAI3 P08754 1/20 0.37
GNAO1 P09471 1/20 0.37
GNAI1 P63096 1/20 0.37
CYP1A2 P05177 1/20 0.31
SPHK1 Q9NYA1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14699799 1.00 GNAI3 (0.37) GNAI3GNAO1GNAI1CYP1A2SPHK1
SCHEMBL15680522 1.00 GNAI3 (0.37) GNAI3GNAO1GNAI1CYP1A2SPHK1
SCHEMBL16111258 1.00 GNAI3 (0.37) GNAI3GNAO1GNAI1CYP1A2SPHK1
SCHEMBL23812547 0.78 CA1 (0.33) GNAI3GNAO1GNAI1CYP1A2
SCHEMBL17052922 0.77
SCHEMBL17052917 0.77
SCHEMBL25962966 0.77
SCHEMBL17053082 0.77
SCHEMBL21780511 0.77
SCHEMBL4168941 0.77 GNAI3 (0.32) GNAI3GNAO1GNAI1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3733663-B1 1-[6-[[4-(PHENYLAMINO)-6-QUINAZOLINYL]OXY]-3-AZABICYCLO[3.1.1]HEPT-3-YL]-2-PROPEN-1-ONE DERIVATIVES AND RELATED COMPOUNDS AS IRREVERSIBLE INHIBITORS OF PAN-HER TYROSINE KINASE FOR THE TREATMENT OF CANCER CHENGDU JINRUI FOUND BIOTECH CO LTD (CN) 2023-05-17 EP disclosed