SCHEMBL2549448

SCHEMBL2549448

CC(=O)C(Cc1ccccc1)Nc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.55
ALDH1A1 P00352 1/20 0.49
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
PAM P19021 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
ALPI P09923 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
XIAP P98170 1/20 0.47
SLC7A5 Q01650 1/20 0.47
TACR1 P25103 1/20 0.47
CTRB1 P17538 3/20 0.46
PPARG P37231 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2722699 0.86 ELANE (0.53) PSMB5ALPIPKMPTGS1XIAP
SCHEMBL1053745 0.86 ELANE (0.53) PSMB5ALPIPKMPTGS1XIAP
SCHEMBL6250861 0.85 PPARG (0.58) PSMB5PPARGCYP1A2
SCHEMBL1533647 0.85 PPARG (0.58) PSMB5PPARGCYP1A2
SCHEMBL1533645 0.85 PPARG (0.58) PSMB5PPARGCYP1A2
SCHEMBL27880853 0.83 ATM (0.60) PSMB5ALDH1A1RAB9AL3MBTL1
SCHEMBL8318346 0.81 TAAR1 (0.52) ALDH1A1CTSSCTSKPAMNPC1
SCHEMBL2628426 0.81 TAAR1 (0.52) ALDH1A1CTSSCTSKPAMNPC1
SCHEMBL17793545 0.81 ALDH1A1 (0.51) ALDH1A1CTSSCTSKPAMNPC1
SCHEMBL28213489 0.81 NAPRT (0.45) PSMB5ALDH1A1NPC1RAB9APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed