SCHEMBL2551450

SCHEMBL2551450

COc1ccc(-n2c(C)nnc2S)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 2/20 0.56
AVPR1A P37288 2/20 0.50
AVPR2 P30518 1/20 0.50
GAA P10253 1/20 0.45
GLA P06280 1/20 0.44
TNKS2 Q9H2K2 3/20 0.44
CYP2C9 P11712 2/20 0.44
TNKS O95271 1/20 0.44
CYP3A4 P08684 1/20 0.44
AXIN2 Q9Y2T1 1/20 0.44
NPC1 O15118 1/20 0.44
CYP1A2 P05177 1/20 0.43
MAPK1 P28482 1/20 0.42
MAPT P10636 2/20 0.41
THRB P10828 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 2/20 0.41
HPGD P15428 1/20 0.41
CUL4A Q13619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11068984 0.91 OXTR (0.52) OXTRAVPR1AAVPR2GAANPC1
SCHEMBL10012186 0.83 OXTR (0.61) OXTRAVPR1AAVPR2GLAHTT
SCHEMBL13703856 0.81 KDM4E (0.47) OXTRAVPR1AGAATNKS2CYP2C9
SCHEMBL6402514 0.79 OXTR (0.57) OXTRAVPR1AAVPR2GLATNKS2
SCHEMBL12110672 0.79 OXTR (0.69) OXTRAVPR1AAVPR2GAAGLA
SCHEMBL11384854 0.78 TLR8 (0.44) OXTRGAAGLACYP2C9CYP3A4
SCHEMBL12110605 0.78 KDM4E (0.46) AVPR1AGAAGLATNKS2NPC1
SCHEMBL11919913 0.78 OXTR (0.52) OXTRAVPR1AAVPR2GAAGLA
SCHEMBL1562739 0.77 AVPR1A (0.56) OXTRAVPR1AGAAMAPK1HTT
SCHEMBL6406225 0.77 OXTR (0.55) OXTRAVPR1AAVPR2GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011122815-A2 NOVEL QUINOXALINE DERIVATIVES DONG-A PHARM.CO.,LTD. (KR) 2011-10-06 WO disclosed
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof AGRIUS GROUP, LLC. 2005-12-29 US disclosed
US-4268680-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1981-05-19 US disclosed
US-4244964-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1981-01-13 US disclosed
US-4232034-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA, N.V. (BE) 1980-11-04 US disclosed
US-4229581-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1980-10-21 US disclosed
US-4229460-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1980-10-21 US disclosed
US-4160841-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA, N.V. (BE) 1979-07-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof ABCG2, ATP5ME, DNTT OXTR 4696/4885AVPR1A 4869/4885AVPR2 4873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.