SCHEMBL25515775

SCHEMBL25515775

Cc1n[nH]c2ccc(-c3nnc(C(F)(F)F)o3)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.48
CDC7 O00311 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
HTR7 P34969 1/20 0.39
JAK2 O60674 2/20 0.38
NOTUM Q6P988 2/20 0.38
TLR8 Q9NR97 2/20 0.37
TLR7 Q9NYK1 2/20 0.37
PIM3 Q86V86 2/20 0.36
PIM2 Q9P1W9 2/20 0.36
MAPK1 P28482 1/20 0.36
MAP2K4 P45985 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
MAPKAPK3 Q16644 1/20 0.36
MAPK6 Q16659 1/20 0.36
TLR9 Q9NR96 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
PIM1 P11309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30408728 1.00 HDAC6 (0.48) HDAC6CDC7CCNE1CDK2DBF4
SCHEMBL25195476 0.82 TLR8 (0.46) CDC7CCNE1CDK2DBF4JAK2
SCHEMBL19321936 0.74 HDAC6 (0.55) HDAC6HTR7NOTUM
SCHEMBL6763933 0.72 HDAC6 (0.55) HDAC6HTR7PIM3PIM2PIM1
SCHEMBL22116919 0.72 NPC1 (0.56) HDAC6MAPK1
SCHEMBL2891668 0.71 HDAC6 (0.51) HDAC6HTR7NOTUM
SCHEMBL13122324 0.70 MAP2K4 (0.56) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6
SCHEMBL30203753 0.70 HPGD (0.63) HDAC6NOTUM
SCHEMBL19317251 0.70 HDAC6 (0.50) HDAC6HTR7NOTUM
SCHEMBL19188029 0.69 JAK2 (0.57) CDC7CDK2JAK2MAPK1MAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078337-A1 CDK8/19 DUAL INHIBITORS AND METHODS OF USE INSILICO MEDICINE IP LIMITED (CN) 2023-05-11 WO disclosed