SCHEMBL2552447

SCHEMBL2552447

CN(C)C#Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.55
NPSR1 Q6W5P4 1/20 0.48
GRM5 P41594 3/20 0.47
KCNH2 Q12809 1/20 0.46
NPC1 O15118 2/20 0.43
MTOR P42345 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 2/20 0.42
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
THPO P40225 1/20 0.41
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
HTR2A P28223 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22326439 0.80 MAPT (0.50) APPNPSR1GRM5KCNH2NPC1
SCHEMBL28389232 0.73 NPC1 (0.48) APPNPSR1GRM5KCNH2NPC1
SCHEMBL13073860 0.73 CYP2A6 (0.61) GRM5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10699281 0.73 APP (0.48) APPNPSR1GRM5KCNH2NPC1
Diphenylacetylene SCHEMBL29188592 0.73 APP (1.00) APPGRM5KCNH2NPC1MTOR
Diphenylacetylene SCHEMBL68254 0.73 APP (1.00) APPGRM5KCNH2NPC1MTOR
Diphenylacetylene SCHEMBL960609 0.73 APP (1.00) APPGRM5KCNH2NPC1MTOR
SCHEMBL497768 0.72 TSHR (0.48) APPNPSR1GRM5KCNH2NPC1
SCHEMBL2923198 0.72 APP (0.52) APPNPSR1GRM5KCNH2NPC1
SCHEMBL22326436 0.72 APP (0.55) APPNPSR1KCNH2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117209452-A Difluoro benzothiadiazole full-color fluorescent molecule, preparation and application thereof 华南师范大学 2023-12-12 CN claimed
EP-3601282-B1 NOVEL PYRIDO[2,3-B]INDOLE COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTION HOFFMANN LA ROCHE (CH) 2021-07-21 EP claimed
EP-1651621-B1 2- (QUINOXALIN-5-YLSULFONYLAMINO) -BENZAMIDE COMPOUNDS AS CCK2 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2008-08-06 EP claimed
CN-117209452-A Difluoro benzothiadiazole full-color fluorescent molecule, preparation and application thereof 华南师范大学 2023-12-12 CN disclosed
CN-111073724-B Lithium-based lubricating grease and preparation method thereof 中国石油化工股份有限公司 2022-08-09 CN disclosed
CN-111100158-B Silole derivative, preparation method and application thereof, and photoluminescent lubricating grease 中国石油化工股份有限公司 2022-07-15 CN disclosed
CN-113754603-A Application of isoxazole compound as viscosity fluorescent probe 浙江工业大学 2021-12-07 CN disclosed
CN-111100158-A Silole derivative, preparation method and application thereof, and photoluminescent lubricating grease 中国石油化工股份有限公司 2020-05-05 CN disclosed
CN-111073724-A Lithium-based lubricating grease and preparation method thereof 中国石油化工股份有限公司 2020-04-28 CN disclosed
CN-111073725-A Photoluminescent grease composition, photoluminescent material and preparation method thereof 中国石油化工股份有限公司 2020-04-28 CN disclosed
CN-105793804-A Method for producing touch sensor member, and touch sensor member 东丽株式会社 2016-07-20 CN disclosed
EP-0776893-B1 Azaheterocyclic compounds having tachykinin receptor antagonist activity; Nk1 and NK2 SANKYO CO (JP) 2002-02-27 EP disclosed
EP-0834499-B1 Process for the preparation of aromatic vinyl compounds DAINIPPON INK & CHEMICALS (JP) 2001-07-25 EP disclosed
US-6159967-A Heterocyclic compounds having tachykinin receptor antagonist activity their preparation and their use SANKYO COMPANY, LIMITED (JP) 2000-12-12 US disclosed
EP-0834499-A1 Process for the preparation of aromatic vinyl compounds DAINIPPON INK AND CHEMICALS, INC. (JP) 1998-04-08 EP disclosed
WO-1997027049-A1 HYPERPOLARIZABLE COMPOUNDS AND DEVICES FABRICATED THEREFROM THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1997-07-31 WO disclosed
EP-0776893-A1 Azaheterocyclic compounds having tachykinin receptor antagonist activity; Nk1 and NK2 SANKYO COMPANY LIMITED (JP) 1997-06-04 EP disclosed
US-3981893-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DT) 1976-09-21 US disclosed
US-3974290-A Vasodilating and antihypertensive compositions and methods of effecting vasodilation and treating hypertension utilizing 2-amino-4H pyrane as the active agent BAYER AKTIENGESELLSCHAFT (DT) 1976-08-10 US disclosed
US-3966767-A CORONARY ACTION, ANTI-HYPERTENSIVE AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed