SCHEMBL25528384

SCHEMBL25528384

COc1nc(N2CCCCC2)ncc1N

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
MEN1 O00255 1/20 0.46
RECQL P46063 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
POLB P06746 1/20 0.43
PIK3CA P42336 2/20 0.40
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
TSHR P16473 2/20 0.39
LMNA P02545 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PTPN11 Q06124 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18690473 0.86 HRH4 (0.50) MEN1KMT2ATSHRALDH1A1HRH4
SCHEMBL25528429 0.84 PIK3CA (0.49) MEN1KMT2ASMN1; SMN2PIK3CATSHR
SCHEMBL28061994 0.82 KMT2A (0.47) HTTMEN1RECQLKMT2AATM
SCHEMBL28827424 0.80 KMT2A (0.44) HTTMEN1RECQLKMT2AATM
SCHEMBL25528278 0.78 PTPN11 (0.36) KCNQ3KCNQ2TSHRALDH1A1PTPN11
SCHEMBL20089101 0.78 PTPN11 (0.48) HTTKMT2ASMN1; SMN2POLBPIK3CA
SCHEMBL1776789 0.75 PTPN11 (0.49) HTTKMT2ASMN1; SMN2POLBPIK3CA
SCHEMBL26647296 0.75 PTPN11 (0.44) HTTMEN1RECQLKMT2AATM
SCHEMBL25528324 0.75 BACE1 (0.33) KCNQ3KCNQ2PTPN11
SCHEMBL27316944 0.75 POLB (0.55) SMN1; SMN2POLBKCNQ3KCNQ2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078411-A1 AZASPIRO COMPOUND 南京明德新药研发有限公司 2023-05-11 WO disclosed