SCHEMBL25528429

SCHEMBL25528429

COc1nc(N2CCOCC2)ncc1N

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.49
MTOR P42345 6/20 0.49
PIK3CD O00329 2/20 0.49
PIK3CB P42338 2/20 0.49
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 1/20 0.48
PIK3R1 P27986 5/20 0.46
MAPK1 P28482 3/20 0.44
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 2/20 0.44
TSHR P16473 2/20 0.44
USP2 O75604 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528384 0.84 HTT (0.46) PIK3CAKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL18690473 0.83 HRH4 (0.50) KMT2AALDH1A1MEN1CYP1A2TSHR
SCHEMBL24158887 0.79 PTPN11 (0.48) PIK3CAMTORPIK3CDKMT2AKDM4E
SCHEMBL5765855 0.79 MAPK1 (0.50) PIK3CAMTORKMT2AKDM4EPIK3R1
SCHEMBL26646893 0.79 PIK3CA (0.55) PIK3CAMTORPIK3CDPIK3CBKMT2A
SCHEMBL10998627 0.76 PIK3CA (0.52) PIK3CAMTORPIK3CDPIK3CBKMT2A
SCHEMBL24158953 0.76 PTPN11 (0.51) PIK3CDKDM4EALDH1A1SMN1; SMN2CYP1A2
SCHEMBL25528278 0.76 PTPN11 (0.36) ALDH1A1TSHRUSP2HSD17B10
SCHEMBL11697780 0.75 KCNQ3 (0.47) PIK3CAMTORKMT2AKDM4EPIK3R1
SCHEMBL2416637 0.74 SMPD3 (0.47) KMT2AKDM4EALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078411-A1 AZASPIRO COMPOUND 南京明德新药研发有限公司 2023-05-11 WO disclosed