SCHEMBL25529316

SCHEMBL25529316

CNc1ncc(C(F)(F)F)c(C)n1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 19/20 0.47
CYP1A2 P05177 9/20 0.47
ULK1 O75385 1/20 0.45
TTK P33981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15221838 0.81 LRRK2 (0.60) LRRK2CYP1A2ULK1
SCHEMBL11916190 0.80 LRRK2 (0.44) LRRK2CYP1A2
SCHEMBL31725453 0.79 AURKA (0.54) LRRK2CYP1A2ULK1
SCHEMBL31725454 0.79 AURKA (0.54) LRRK2CYP1A2ULK1
SCHEMBL12149236 0.79 LRRK2 (0.47) LRRK2CYP1A2ULK1
SCHEMBL25529238 0.77 ULK1 (0.45) LRRK2CYP1A2ULK1
SCHEMBL10297751 0.75 LRRK2 (0.35) LRRK2CYP1A2ULK1TTK
SCHEMBL21184419 0.75 ULK1 (0.67) ULK1
SCHEMBL12688604 0.75 LRRK2 (0.38) LRRK2CYP1A2ULK1TTK
SCHEMBL14621356 0.74 ULK1 (0.61) ULK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed