SCHEMBL25530684

SCHEMBL25530684

CN1CCC(CNC(=O)c2cccc(CN(CC=O)C(=O)c3ccc(-c4ccnc(N)c4)cc3N(C)C)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.43
MAP4K4 O95819 2/20 0.42
PARP1 P09874 1/20 0.42
GLS O94925 2/20 0.37
MAPK14 Q16539 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
KCNH2 Q12809 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25530669 0.83 AOC3 (0.36) ROCK2ROCK1
SCHEMBL25530657 0.82 ROCK2 (0.38) ROCK2ROCK1GSK3B
SCHEMBL25531248 0.73 ROCK2 (0.40) ROCK2MAPK14PIK3C3KCNH2IRAK4
SCHEMBL25528649 0.70 ROCK2 (0.44) ROCK2MAP4K4PARP1GLSMAPK14
SCHEMBL25528196 0.70 ROCK2 (0.43) ROCK2MAP4K4PARP1GLSMAPK14
SCHEMBL25530636 0.69 ROCK2 (0.43) ROCK2MAP4K4PARP1GLSMAPK14
SCHEMBL25528744 0.69 ROCK2 (0.46) ROCK2MAP4K4PARP1GLSMAPK14
SCHEMBL25529530 0.69 ROCK2 (0.41) ROCK2ROCK1
SCHEMBL25718992 0.68 ROCK2 (0.71) ROCK2MAP4K4ROCK1GSK3B
SCHEMBL20113313 0.66 ROCK2 (0.58) ROCK2PARP1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed