SCHEMBL2553597

SCHEMBL2553597

CCOC(=O)C(c1ccccc1C(F)(F)F)N(C)C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 1/20 0.43
POLQ O75417 1/20 0.42
EPHX2 P34913 5/20 0.41
PPARG P37231 4/20 0.41
CNR2 P34972 2/20 0.41
KMT2A Q03164 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
ACP3 P15309 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
PIN1 Q13526 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915633 0.82 CNR2 (0.43) KDM4EALDH1A1POLQCNR2KMT2A
SCHEMBL29268488 0.81 EPHX2 (0.46) KDM4EALDH1A1EPHX2PPARGCNR2
SCHEMBL2550492 0.80 TDP1 (0.43) KDM4EALDH1A1KMT2ASLC6A2SLC6A4
SCHEMBL753073 0.80 POLQ (0.47) POLQPPARGCNR2ACP3
SCHEMBL8921824 0.80 ACP3 (0.43) ALDH1A1POLQCNR2ACP3POLB
SCHEMBL6929206 0.79 KDM4E (0.44) KDM4EALDH1A1EPHX2PPARGCNR2
SCHEMBL2550711 0.79 PIN1 (0.41) KDM4EALDH1A1KMT2ASLC6A2SLC6A4
SCHEMBL888787 0.78 POLQ (0.41) ALDH1A1POLQCNR2SLC6A2SLC6A4
SCHEMBL8907146 0.78 ACP3 (0.41) ALDH1A1POLQCNR2ACP3POLB
SCHEMBL167566 0.77 EPHX2 (0.44) KDM4EALDH1A1EPHX2PPARGCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed