SCHEMBL2554328

SCHEMBL2554328

COc1ccccc1C(=O)CC=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.58
CTSD P07339 1/20 0.54
ALDH1A1 P00352 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CTNNB1 P35222 3/20 0.51
WNT3A P56704 3/20 0.51
IDO1 P14902 1/20 0.51
TDO2 P48775 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC1 Q13547 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.50
LMNA P02545 2/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HPGD P15428 2/20 0.47
TP53 P04637 1/20 0.47
GLA P06280 1/20 0.47
STAT3 P40763 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9642042 0.86 NPC1 (0.58) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL31413027 0.83 CTNNB1 (0.56) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL19287106 0.83 CTNNB1 (0.56) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL2554727 0.83 HCRTR1 (0.59) ALDH1A1KMT2AHTTL3MBTL1LMNA
SCHEMBL31413029 0.83 CTNNB1 (0.56) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL15979734 0.81 CTNNB1 (0.71) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL21128714 0.81 NPC1 (0.83) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL29987209 0.81 NPC1 (0.83) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL22118761 0.80 HDAC8 (0.61) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL3702934 0.79 NPC1 (0.64) NPC1CTSDALDH1A1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117466817-A Preparation method of polysubstituted pyrazole derivative 华侨大学 2024-01-30 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-115093323-A Beta-functionalized chiral homoallyl alcohol derivative and preparation method and application thereof 武汉大学 2022-09-23 CN disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
CN-105503635-B A kind of preparation method of the Dicarbonyl derivatives of 2 amido formacyl 1,3 苏州大学 2017-10-10 CN disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed