SCHEMBL3702934

SCHEMBL3702934

COc1ccccc1C(=O)C[O]

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.64
CTSD P07339 1/20 0.59
ALDH1A1 P00352 2/20 0.57
KMT2A Q03164 2/20 0.57
HTT P42858 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
CTNNB1 P35222 3/20 0.55
WNT3A P56704 3/20 0.55
IDO1 P14902 1/20 0.55
TDO2 P48775 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC1 Q13547 1/20 0.55
LMNA P02545 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HPGD P15428 2/20 0.51
STAT3 P40763 1/20 0.51
TP53 P04637 1/20 0.51
GLA P06280 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28199327 0.86 NPC1 (0.62) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL21128714 0.86 NPC1 (0.83) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL29987209 0.86 NPC1 (0.83) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL15979734 0.86 CTNNB1 (0.71) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL878658 0.84 NPC1 (0.64) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL1448202 0.84 NPC1 (0.64) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL29738645 0.84 NPC1 (0.64) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL6488893 0.82 NPC1 (0.62) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL598461 0.82 L3MBTL1 (0.64) NPC1CTSDALDH1A1KMT2AHTT
SCHEMBL18907831 0.82 NPC1 (0.62) NPC1CTSDALDH1A1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123441-B1 VINCALEUKOBLASTINE DERIVATIVES LILLY INDUSTRIES LIMITED (GB) 1990-10-03 EP claimed
US-4675400-A FORM CONJUGATES WITH IMMUNOGLOBULINS; ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1987-06-23 US claimed
US-4596676-A Bifunctional ester derivatives of 4-desacetyl indole-dihydroindole alkaloids LILLY INDUSTRIES LIMITED (GB) 1986-06-24 US claimed
EP-0123441-A1 Vincaleukoblastine derivatives LILLY INDUSTRIES LIMITED (GB) 1984-10-31 EP claimed
EP-2396017-A1 APOLIPOPROTEIN A-I MIMICS Cerenis Therapeutics SA (FR) 2011-12-21 EP disclosed
WO-2010093918-A1 APOLIPOPROTEIN A-I MIMICS CERENIS THERAPEUTICS SA (FR) 2010-08-19 WO disclosed
EP-0686636-B1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA CO (JP) 2001-04-04 EP disclosed
US-5840895-A INTERMEDIATES FOR ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5686442-A ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1997-11-11 US disclosed
EP-0686636-A1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-12-13 EP disclosed
EP-0123441-B1 VINCALEUKOBLASTINE DERIVATIVES LILLY INDUSTRIES LIMITED (GB) 1990-10-03 EP disclosed
US-4675400-A FORM CONJUGATES WITH IMMUNOGLOBULINS; ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1987-06-23 US disclosed
US-4596676-A Bifunctional ester derivatives of 4-desacetyl indole-dihydroindole alkaloids LILLY INDUSTRIES LIMITED (GB) 1986-06-24 US disclosed
EP-0123441-A1 Vincaleukoblastine derivatives LILLY INDUSTRIES LIMITED (GB) 1984-10-31 EP disclosed