SCHEMBL2554561

SCHEMBL2554561

COC(=O)C(Br)C1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.47
ALDH1A1 P00352 3/20 0.45
NPSR1 Q6W5P4 3/20 0.45
THRB P10828 1/20 0.44
TSHR P16473 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
SLC6A3 Q01959 2/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
MMP2 P08253 2/20 0.39
CA9 Q16790 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1605366 0.98 TP53 (0.50) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL20740436 0.98 TP53 (0.50) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL14218540 0.98 TP53 (0.50) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL31572346 0.96 THRB (0.44) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL15618893 0.91
SCHEMBL4491334 0.82 THRB (0.61) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL5268464 0.82 SLC6A2 (0.44) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL1605421 0.82 MEN1 (0.36) TP53ALDH1A1NPSR1THRBTSHR
SCHEMBL10066711 0.80 TP53 (0.50) TP53ALDH1A1NPSR1THRBKMT2A
SCHEMBL19941727 0.80 TP53 (0.62) TP53ALDH1A1NPSR1THRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
EP-0045165-B1 RHODANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION, AND ALDOSE REDUCTASE INHIBITORS CONTAINING SUCH DERIVATIVES ONO PHARMACEUTICAL CO., LTD. (JP) 1986-03-12 EP disclosed
US-4446143-A Rhodanine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1984-05-01 US disclosed
EP-0045165-A1 Rhodanine derivatives, a process for their preparation, and aldose reductase inhibitors containing such derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1982-02-03 EP disclosed