SCHEMBL25549

SCHEMBL25549

COCCOC(=O)C1=C(C)NC(C)=C(COC/C=C/c2ccccc2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 8/20 0.83
MEN1 O00255 6/20 0.83
KMT2A Q03164 6/20 0.83
CACNA1B Q00975 3/20 0.83
ADORA3 P0DMS8 2/20 0.83
MLNR O43193 1/20 0.83
NR1I2 O75469 1/20 0.83
CACNA1H O95180 1/20 0.83
NR3C1 P04150 1/20 0.83
TBXA2R P21731 1/20 0.83
HTT P42858 1/20 0.83
PDE4D Q08499 1/20 0.83
SLC29A1 Q99808 1/20 0.83
CYP1A2 P05177 4/20 0.64
CYP3A4 P08684 4/20 0.64
CYP2C9 P11712 4/20 0.64
CYP2C19 P33261 4/20 0.64
MAPT P10636 4/20 0.64
LMNA P02545 3/20 0.64
CYP2D6 P10635 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cilnidipine SCHEMBL25551 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL29367885 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL31398437 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL25550 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL30209784 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL3334757 0.91 CACNA1C (1.00) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL28356318 0.90 CACNA1C (0.98) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL29248832 0.90 CACNA1C (0.98) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL27852253 0.89 CACNA1C (0.95) CACNA1CMEN1KMT2ACACNA1BADORA3
Cilnidipine SCHEMBL29141421 0.86 CACNA1C (0.90) CACNA1CMEN1KMT2ACACNA1BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5876 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4741492-A2 NECROSIS INHIBITOR Linkgevity Limited (GB) 2026-05-13 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
WO-2026090605-A2 COMPOSITIONS AND METHODS COMPRISING TARGETED LIPOSOMAL THERAPEUTIC VACCINES DREXEL UNIVERSITY (US) 2026-04-30 WO claimed
EP-4691462-A1 SILYBIN-CONTAINING COMPOSITION Tianjin Tasly Sants Pharmaceutical Co., Ltd. (CN) 2026-02-11 EP claimed
EP-4683634-A1 TREATMENT OF SCLERODERMA Aisa Pharma, Inc. (US) 2026-01-28 EP claimed
EP-4648769-A2 NECROSIS INHIBITOR Linkgevity Limited (GB) 2025-11-19 EP claimed
US-20250345332-A1 APROCITENTAN FOR THE TREATMENT OF HYPERTENSION IDORSIA PHARMACEUTICALS LTD (CH) 2025-11-13 US claimed
US-12441687-B2 Drp1-filamin complex formation inhibitors Rdiscovery, LLC (US) 2025-10-14 US claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
EP-4615577-A1 METHODS OF TREATING EYE PAIN AND EYE DISORDERS Aisa Pharma, Inc. (US) 2025-09-17 EP claimed
EP-1303305-A2 EPOXY-STEROIDAL ALDOSTERONE ANTAGONIST AND CALCIUM CHANNEL BLOCKER COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE Pharmacia Corporation (US) 2003-04-23 EP claimed
US-20030073127-A1 NOVEL CALCIUM CHANNEL DRUGS AND USES THERAVANCE BIOPHARMA R&D IP, LLC 2003-04-17 US claimed
US-20030073670-A1 Stabilized pharmaceutical compositions containing a calcium channel blocker SANKYO COMPANY, LIMITED (JP) 2003-04-17 US claimed
WO-2002087556-A9 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS INC (US) 2003-03-20 WO claimed
US-20030055027-A1 Epoxy-steroidal aldosterone antagonist and calcium channel blocker combination therapy for treatment of congestive heart failure G. D. SEARLE & CO. (US) 2003-03-20 US claimed
EP-1285655-A1 STABILIZED PHARMACEUTICAL COMPOSITIONS CONTAINING CALCIUM CHANNEL BLOCKERS Sankyo Company, Limited (JP) 2003-02-26 EP claimed
WO-2002087556-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS, INC. (US) 2002-11-07 WO claimed
WO-2002060461-A1 BLOOD BRAIN BARRIER MODULATION USING STRESSED AUTOLOGOUS BLOOD CELLS VASOGEN IRELAND LIMITED (IE) 2002-08-08 WO claimed
US-20020042405-A1 Epoxy-steroidal aldosterone antagonist and calcium channel blocker combination therapy for treatment of congestive heart failure SCHUH JOSEPH R (US) 2002-04-11 US claimed
WO-2002009761-A2 EPOXY-STEROIDAL ALDOSTERONE ANTAGONIST AND CALCIUM CHANNEL BLOCKER COMBINATION THERAPY FOR TREATMENT OF CONGESTIVE HEART FAILURE PHARMACIA CORPORATION (US) 2002-02-07 WO claimed