SCHEMBL25555209

SCHEMBL25555209

COCCN(C)c1cc(Oc2cc(C#N)ccc2-c2ncc(CN)cn2)n(C)n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 5/20 0.35
EGLN1 Q9GZT9 3/20 0.34
FASN P49327 5/20 0.33
ADORA2A P29274 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
ADK P55263 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
USP1 O94782 1/20 0.31
PRKDC P78527 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25555153 0.93 EGLN1 (0.33) NSD2EGLN1FASNADORA2AHCRTR1
SCHEMBL25555210 0.90 NSD2 (0.35) NSD2EGLN1FASNADORA2AHCRTR1
SCHEMBL25555213 0.88 EGLN1 (0.37) EGLN1ADORA2AHCRTR1HCRTR2CYP19A1
SCHEMBL25554934 0.88 NSD2 (0.36) NSD2CYP19A1CYP11B1CYP11B2PRKDC
SCHEMBL25555255 0.88 EGLN1 (0.35) EGLN1ADORA2ACYP19A1CYP11B1CYP11B2
SCHEMBL25555317 0.87 NSD2 (0.33) NSD2
SCHEMBL30257251 0.87 NSD2 (0.33) NSD2
SCHEMBL25555309 0.86 NSD2 (0.34) NSD2PRKDC
SCHEMBL25058268 0.85 HCRTR1 (0.32) NSD2HCRTR1HCRTR2CYP19A1CYP11B1
SCHEMBL25554975 0.85 NSD2 (0.37) NSD2CYP19A1CYP11B1CYP11B2PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2023-06-01 US disclosed
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2023-06-01 US disclosed
EP-4137481-A1 ARYL OR HETEROARYL DERIVATIVE Teijin Pharma Limited (JP) 2023-02-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230167073-A1 ARYL OR HETEROARYL DERIVATIVE ARRB1, NR3C2, TRPC6 NSD2 3265/4885EGLN1 3878/4885FASN 4505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.