SCHEMBL25561920

SCHEMBL25561920

CN1CCN(c2ccc(Nc3nc(NC4CCOCC4)c(-c4ccccc4C(N)=O)nc3C(N)=O)cc2)CC1

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EML4 Q9HC35 11/20 0.73
ALK Q9UM73 11/20 0.73
RET P07949 16/20 0.72
ROS1 P08922 16/20 0.72
FLT3 P36888 16/20 0.72
SYK P43405 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25562169 0.88 EML4 (0.70) EML4ALKRETROS1FLT3
SCHEMBL25562019 0.86 RET (0.74) EML4ALKRETROS1FLT3
SCHEMBL25562018 0.86 RET (0.75) EML4ALKRETROS1FLT3
SCHEMBL25561959 0.86 RET (0.74) EML4ALKRETROS1FLT3
SCHEMBL25562853 0.86 RET (0.74) EML4ALKRETROS1FLT3
SCHEMBL25562047 0.86 EML4 (0.73) EML4ALKRETROS1FLT3
SCHEMBL25561960 0.86 RET (0.73) EML4ALKRETROS1FLT3
SCHEMBL25562194 0.85 EML4 (0.69) EML4ALKRETROS1FLT3
SCHEMBL25561929 0.85 FLT3 (0.72) EML4ALKRETROS1FLT3
SCHEMBL25562123 0.84 EML4 (0.70) EML4ALKRETROS1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230167099-A1 NEW PYRAZINE COMPOUND Wigen Biomedicine Technology (shanghai) Co., Ltd. (CN) 2023-06-01 US disclosed
US-20230167099-A1 NEW PYRAZINE COMPOUND Wigen Biomedicine Technology (shanghai) Co., Ltd. (CN) 2023-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230167099-A1 NEW PYRAZINE COMPOUND EGFR, ERBB2, WEE1 EML4 163/4885ALK 131/4885RET 22/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.