SCHEMBL2556366

SCHEMBL2556366

CCc1nn(-c2ccc(F)cc2)c(C)c1OC(=O)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDE4D Q08499 3/20 0.40
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TP53 P04637 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2561878 0.83 PDE4D (0.41) L3MBTL1ALDH1A1PDE4DPDE4APDE4B
SCHEMBL12264390 0.83 PDE4D (0.52) MAPTTDP1L3MBTL1ALDH1A1NPSR1
SCHEMBL2553638 0.80 PDE4A (0.38) ALDH1A1NPSR1PDE4DPDE4APDE4B
SCHEMBL2576433 0.78 TSHR (0.47) MAPTL3MBTL1ALDH1A1NPSR1PDE4D
SCHEMBL14482912 0.71 MEN1 (0.47) ALDH1A1NPSR1PDE4DPDE4APDE4B
SCHEMBL2563146 0.71 ALDH1A1 (0.52) MAPTALDH1A1NPSR1PDE4DTSHR
SCHEMBL2555825 0.70 PDE4D (0.63) MAPTTDP1ALDH1A1NPSR1PDE4D
SCHEMBL30929673 0.70 ALDH1A1 (0.55) MAPTTDP1L3MBTL1ALDH1A1MEN1
SCHEMBL2560863 0.70 ALDH1A1 (0.55) ALDH1A1NPSR1MEN1KMT2ASMN1; SMN2
SCHEMBL12264383 0.69 PDE4D (0.47) L3MBTL1ALDH1A1NPSR1PDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed