SCHEMBL2556578

SCHEMBL2556578

Cc1ccccc1-c1ncccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 8/20 0.58
CYP3A4 P08684 7/20 0.58
CYP2C19 P33261 6/20 0.58
GAA P10253 3/20 0.50
CYP2D6 P10635 4/20 0.49
HSD17B10 Q99714 4/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
ALOX15 P16050 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
MITF O75030 1/20 0.49
PKM P14618 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
ALDH1A1 P00352 5/20 0.47
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21742567 0.91 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL21742862 0.82 SLC6A7 (0.49) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL27018672 0.82 BRD4 (0.44) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL16806048 0.81 CYP1A2 (0.42) CYP1A2CYP3A4CYP2C19GAANPC1
SCHEMBL9444918 0.81 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL10599951 0.81 KDM4E (0.45) CYP1A2CYP3A4GAACYP2D6NPC1
SCHEMBL28133533 0.81 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL8365591 0.81 CYP1A2 (0.64) CYP1A2CYP3A4CYP2C19GAACYP2D6
SCHEMBL13531392 0.79 GAA (0.46) CYP1A2CYP3A4CYP2C19GAACYP2D6
Ammonia Solution, Strong SCHEMBL27685788 0.79 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C19GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102238950-B Certain kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use CHDI FOUNDATION INC (US) 2014-05-07 CN claimed
CN-102238950-A Certain kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use CHDI INC (US) 2011-11-09 CN claimed
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN claimed
CN-1324015-C Pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2007-07-04 CN claimed
CN-1630644-A Novel pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2005-06-22 CN claimed
US-11825734-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-11-21 US disclosed
WO-2021222614-A1 INHIBITOR OF APOPTOSIS (IAP) PROTEIN ANTAGONISTS Sanford Burnham Prebys Medical Discovery Institute (US) 2021-11-04 WO disclosed
WO-2020065614-A1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2020-04-02 WO disclosed
US-9905777-B2 Compound and organic electroluminescence device comprising same DOOSAN CORPORATION (KR) 2018-02-27 US disclosed
US-9905777-B2 Compound and organic electroluminescence device comprising same DOOSAN CORPORATION (KR) 2018-02-27 US disclosed
WO-2018033082-A1 INHIBITORS OF INFLUENZA VIRUS REPLICATION, APPLICATION METHODS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2018-02-22 WO disclosed
WO-2017209487-A1 ORGANIC COMPOUND AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING SAME 주식회사 두산 2017-12-07 WO disclosed
CN-1324015-C Pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2007-07-04 CN disclosed
WO-2006127948-A2 N-TERMINALLY MODIFIED GLP-1 RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-11-30 WO disclosed
CN-1630644-A Novel pyridine and pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2005-06-22 CN disclosed
US-H890-H Herbicidal heterocyclicbenzylsulfonamides Rorer, Morris P. (US) 1991-02-05 US disclosed
US-4859670-A 2-Azolylmethyl-2-aryl-1,3-dioxolanes and the salts thereof, agents containing same, and the use thereof HOECHST AKTIENGESELLSCHAFT (DE) 1989-08-22 US disclosed
US-4699649-A Herbicidal heterocyclicbenzylsulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-10-13 US disclosed
EP-0237962-A2 2-Azolylmethyl-2-aryl-1,3-dioxolanes and their preparation, compositions containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-09-23 EP disclosed
EP-0164268-A2 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-12-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11825734-B2 Organic electroluminescent materials and devices OCIAD2, OCIAD1, OSBP CYP1A2 1592/4885CYP3A4 523/4885CYP2C19 1450/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.