SCHEMBL2559530

SCHEMBL2559530

CN(C)c1cccc(-c2cnc(N3CCCCC3)nc2)c1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 10/20 0.55
DHFR P00374 1/20 0.44
FYN P06241 7/20 0.43
GRIN1 Q05586 1/20 0.41
GRIN2B Q13224 1/20 0.41
NTRK1 P04629 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2557199 0.82 BRAF (0.43) AOC3FYN
SCHEMBL13606215 0.81 AOC3 (0.52) AOC3DHFRGRIN2B
SCHEMBL2554399 0.79 SMN1; SMN2 (0.61) AOC3FYN
SCHEMBL13680656 0.79 AOC3 (0.51) AOC3DHFRGRIN2B
SCHEMBL2553959 0.79 HRH4 (0.43)
SCHEMBL2559391 0.79 PIK3CA (0.51)
SCHEMBL19496719 0.78 AOC3 (0.69) AOC3
SCHEMBL13606217 0.78 CNR2 (0.51) AOC3DHFR
SCHEMBL13606218 0.77 AOC3 (0.50) AOC3DHFR
SCHEMBL13606216 0.77 KDM4E (0.56) AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011130515-A1 ARYLTHIAZOLYL PIPERIDINES AND RELATED COMPOUNDS AS MODULATORS OF SURVIVAL MOTOR NEURON (SMN) PROTEIN PRODUCTION THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-10-20 WO disclosed