SCHEMBL25600216

SCHEMBL25600216

Cc1noc2c3c(ccc12)CN(CC1CCNCC1)CC3

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.40
DRD3 P35462 1/20 0.40
KDM2B Q8NHM5 1/20 0.38
HRH3 Q9Y5N1 3/20 0.34
BRD4 O60885 1/20 0.34
PDE1B Q01064 1/20 0.33
PIK3R1 P27986 2/20 0.32
PIK3CA P42336 2/20 0.32
DRD1 P21728 1/20 0.32
DRD5 P21918 1/20 0.32
FAAH O00519 1/20 0.32
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 1/20 0.31
HIF1A Q16665 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CACNA2D1 P54289 1/20 0.30
CACNA1B Q00975 1/20 0.30
CACNB1 Q02641 1/20 0.30
HTR7 P34969 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25600646 0.92 HRH1 (0.44) HRH1DRD3KDM2BHRH3BRD4
SCHEMBL25600320 0.80 HRH1 (0.45) HRH1DRD3KDM2BHRH3BRD4
SCHEMBL25593050 0.80 HRH1 (0.46) HRH1DRD3HRH3
SCHEMBL25595129 0.79 KDM2B (0.35) HRH1DRD3KDM2B
SCHEMBL25595528 0.77 BCHE (0.32)
SCHEMBL25600571 0.76 SSTR4 (0.33)
SCHEMBL25595529 0.75 KHK (0.34) HRH1DRD3CYP1A2CYP3A4HIF1A
SCHEMBL25595530 0.74 HRH1 (0.36) HRH1DRD3HRH3BRD4CYP1A2
SCHEMBL25592128 0.73 DRD3 (0.43) HRH1DRD3BRD4DRD5CYP1A2
SCHEMBL25595531 0.72 KDM2B (0.43) HRH1DRD3KDM2BBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed