SCHEMBL25604136

SCHEMBL25604136

CC(=O)Oc1ccc2c(c1)CN(C(=O)C(F)(F)F)C2

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.60
ESR2 Q92731 3/20 0.60
ABHD6 Q9BV23 12/20 0.46
MGLL Q99685 5/20 0.46
PKM P14618 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
OPRM1 P35372 1/20 0.41
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25825941 0.85 ESR1 (0.80) ESR1ESR2ABHD6MGLL
SCHEMBL31670368 0.78 HDAC6 (0.55) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL7277197 0.76 NOTUM (0.53) ESR1ESR2ABHD6MGLL
SCHEMBL4727849 0.76 ABHD6 (0.58) ESR1ESR2ABHD6MGLL
SCHEMBL10214641 0.75 HDAC6 (0.56) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL29100405 0.75 NOTUM (0.58) ESR1ESR2ABHD6
SCHEMBL25604135 0.75 ESR2 (0.77) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL3895230 0.75 ESR1 (1.00) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL31164691 0.75 ESR1 (0.90) ESR1ESR2ABHD6PKM
SCHEMBL25604095 0.75 ABHD6 (0.54) ESR1ESR2ABHD6ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed