SCHEMBL25604192

SCHEMBL25604192

O=C(N1CCc2cccc(O)c2C1)C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.56
ESR2 Q92731 5/20 0.56
ABHD6 Q9BV23 5/20 0.50
DRD1 P21728 2/20 0.43
DRD3 P35462 2/20 0.43
DRD2 P14416 1/20 0.43
DRD5 P21918 1/20 0.43
EP300 Q09472 1/20 0.42
CREBBP Q92793 1/20 0.42
BCL2L1 Q07817 1/20 0.41
BAD Q92934 1/20 0.41
NOTUM Q6P988 1/20 0.40
HTR5A P47898 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506963 0.90 ESR1 (0.50) ESR1ESR2ABHD6DRD1DRD3
SCHEMBL8177222 0.88 ESR1 (0.56) ESR1ESR2ABHD6BCL2L1BAD
SCHEMBL25825897 0.86 ABHD6 (0.47) ESR1ESR2ABHD6BCL2L1BAD
SCHEMBL587897 0.84 ABHD6 (0.69) ESR1ESR2ABHD6DRD2EP300
SCHEMBL17130540 0.84 ESR1 (0.55) ESR1ESR2ABHD6DRD2EP300
SCHEMBL3885156 0.84 ESR1 (0.51) ESR1ESR2ABHD6DRD2EP300
SCHEMBL19582436 0.83 ESR1 (0.50) ESR1ESR2ABHD6DRD1DRD2
SCHEMBL9913538 0.82 ESR1 (0.49) ESR1ESR2ABHD6EP300CREBBP
SCHEMBL16269409 0.81 DRD1 (0.47) ABHD6DRD1DRD3DRD2DRD5
SCHEMBL9913535 0.81 ABHD6 (0.49) ESR1ESR2ABHD6EP300CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed