SCHEMBL2560944

SCHEMBL2560944

O=C(Nc1ccc2[nH]nc(I)c2c1)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.67
ROCK1 Q13464 4/20 0.67
CCR2 P41597 1/20 0.53
ACKR3 P25106 1/20 0.52
CTNNB1 P35222 5/20 0.51
TCF7L2 Q9NQB0 5/20 0.51
ULK1 O75385 2/20 0.50
WNT1 P04628 1/20 0.49
DYRK1A Q13627 1/20 0.49
LTA4H P09960 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2861604 0.81 MAPK10 (0.67) ROCK2ROCK1CCR2ACKR3CTNNB1
SCHEMBL15022646 0.81 ROCK2 (0.68) ROCK2ROCK1CCR2
SCHEMBL15021912 0.81 ROCK2 (0.68) ROCK2ROCK1CCR2
SCHEMBL12282076 0.80 TTK (0.66) ROCK2ROCK1
SCHEMBL2571386 0.80 ROCK2 (1.00) ROCK2ROCK1CCR2ULK1
Hydrochloric Acid SCHEMBL2568328 0.79 TTK (0.65) ROCK2ROCK1
SCHEMBL2866839 0.77 ROCK2 (0.55) ROCK2ROCK1CCR2ACKR3ULK1
SCHEMBL15021797 0.75 ROCK2 (0.66) ROCK2ROCK1CCR2
SCHEMBL17311705 0.74 ROCK2 (1.00) ROCK2ROCK1
SCHEMBL1554194 0.74 TDP1 (0.61) ROCK2ROCK1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed