SCHEMBL2561886

SCHEMBL2561886

CC1(C)Cc2ccc(NCc3ccc(Br)cn3)cc2C2(COC(NC(=O)OC(C)(C)C)=N2)C1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.36
APP P05067 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
CTSD P07339 4/20 0.33
RORC P51449 1/20 0.32
MAPKAPK2 P49137 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2557900 0.89 BACE1 (0.36) BACE1APPCYP3A4CYP2D6CYP2C9
SCHEMBL449162 0.87 BACE1 (0.46) BACE1APPCYP3A4CYP2D6CYP2C9
SCHEMBL2566485 0.84 BACE1 (0.36) BACE1APPCTSDMAPKAPK2
SCHEMBL447340 0.84 BACE1 (0.45) BACE1CYP3A4CYP2C9CTSD
SCHEMBL446250 0.78 BACE1 (0.42) BACE1CTSD
SCHEMBL447030 0.75 BACE1 (0.49) BACE1APPCYP3A4CYP2D6CYP2C9
SCHEMBL446897 0.71 BACE1 (0.43) BACE1APPCTSD
SCHEMBL450426 0.71 BACE1 (0.45) BACE1APPCYP3A4CYP2D6CYP2C9
SCHEMBL447848 0.70 BACE1 (0.59) BACE1APPCYP3A4CYP2D6CYP2C9
SCHEMBL15264508 0.67 BACE1 (0.67) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123674-A1 COMPOUNDS FOR TREATING NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2011-10-06 WO disclosed