SCHEMBL2564293

SCHEMBL2564293

O=C(O)CCSc1nc2cc[nH]c2c(=O)n1-c1ccc(OCC(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 1/20 0.51
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
NPC1 O15118 1/20 0.41
MAPK1 P28482 1/20 0.39
AR P10275 1/20 0.38
LMNA P02545 2/20 0.37
PIK3CD O00329 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
PIK3CA P42336 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36
TP53 P04637 3/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2564109 0.95 FADS1 (0.50) FADS1MEN1KMT2ANPC1LMNA
SCHEMBL2559985 0.90 FADS1 (0.51) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2991104 0.89 FADS1 (0.50) FADS1MEN1KMT2ANPC1LMNA
SCHEMBL2575941 0.89 FADS1 (0.51) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2565491 0.88 FADS1 (0.53) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2566541 0.88 FADS1 (0.50) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2564675 0.88 KMT2A (0.48) MEN1KMT2ALMNAALDH1A1TP53
SCHEMBL2562601 0.88 FADS1 (0.51) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2566331 0.87 FADS1 (0.49) FADS1MEN1KMT2ALMNAPIK3CD
SCHEMBL2561318 0.87 FADS1 (0.50) FADS1MEN1KMT2ALMNAPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2382218-A1 DELTA-5-DESATURASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-11-02 EP disclosed
WO-2010087467-A1 DELTA-5-DESATURASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-05 WO disclosed