SCHEMBL2564464

SCHEMBL2564464

Brc1ccc(I)c(C=Cc2cc(Br)ccc2I)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.40
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2A6 P11509 3/20 0.33
CASP1 P29466 1/20 0.32
ALOX15 P16050 1/20 0.32
AHR P35869 1/20 0.32
PTPN1 P18031 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MAPT P10636 1/20 0.31
HSP90AA1 P07900 1/20 0.31
TLR9 Q9NR96 1/20 0.31
S100A4 P26447 1/20 0.31
MAPK1 P28482 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2564460 1.00 ERN1 (0.40) ERN1CA12CA9MEN1KMT2A
SCHEMBL14416446 0.82 HPGD (0.35) ERN1CA12CA9MEN1KMT2A
SCHEMBL16955573 0.81 ERN1 (0.42) ERN1CA12CA9MEN1KMT2A
SCHEMBL16956615 0.81 ERN1 (0.38) ERN1CA12CA9CYP2A6CASP1
SCHEMBL137546 0.81 ERN1 (0.57) ERN1CA12CA9MEN1KMT2A
SCHEMBL2584464 0.80 CYP2A6 (0.40) ERN1CA12CA9CYP2A6ALOX15
SCHEMBL14736145 0.80 CYP2A6 (0.40) ERN1CA12CA9CYP2A6ALOX15
SCHEMBL2584466 0.80 CYP2A6 (0.40) ERN1CA12CA9CYP2A6ALOX15
SCHEMBL15452345 0.76 HPGD (0.37) ERN1MEN1KMT2ACASP1KDM4E
SCHEMBL29645435 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130059996-A1 Boron-Containing PI-Electron Materials Incorporating Formally Aromatic and Neutral Borepin Rings THE JOHNS HOPKINS UNIVERSITY 2013-03-07 US disclosed
WO-2011127383-A2 BORON-CONTAINING PI-ELECTRON MATERIALS INCORPORATING FORMALLY AROMATIC AND NEUTRAL BOREPIN RINGS THE JOHNS HOPKINS UNIVERSITY (US) 2011-10-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130059996-A1 Boron-Containing PI-Electron Materials Incorporating Formally Aromatic and Neutral Borepin Rings PNN, CIAPIN1, VNN1 ERN1 1084/4885CA12 904/4885CA9 3464/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.