SCHEMBL2564538

SCHEMBL2564538

O=C1CC2CNCCN2c2cc(OCC3CC3)ccc2N1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.49
CREBBP Q92793 2/20 0.49
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
DRD2 P14416 1/20 0.42
HTR2C P28335 11/20 0.40
HTR2B P41595 6/20 0.40
HTR2A P28223 6/20 0.40
PARP15 Q460N3 1/20 0.39
PARP10 Q53GL7 1/20 0.39
HTR6 P50406 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 1/20 0.38
CYP2D6 P10635 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HTR3A P46098 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAP2K1 Q02750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2021614 1.00 BRD4 (0.49) BRD4CREBBPMAOAMAOBDRD2
SCHEMBL691343 0.87 HTR2C (0.47) HTR2CHTR2BHTR2AHTR6
SCHEMBL2015193 0.87 HTR2C (0.47) HTR2CHTR2BHTR2AHTR6
SCHEMBL2014689 0.83 CREBBP (0.53) BRD4CREBBPMAOAMAOBSLC6A2
SCHEMBL693191 0.83 HTR2C (0.58) MAOAMAOBHTR2CHTR2BHTR2A
SCHEMBL691878 0.83 HTR2C (0.58) MAOAMAOBHTR2CHTR2BHTR2A
SCHEMBL2014698 0.82 CREBBP (0.52) BRD4CREBBPMAOAMAOBHTR2C
SCHEMBL2019541 0.81 HTR2C (0.42) HTR2CHTR2BHTR2AHTR6
SCHEMBL693785 0.80 HTR1A (0.43) CREBBPMAOBDRD2HTR2CHTR2B
SCHEMBL693335 0.79 MAOB (0.46) CREBBPMAOAMAOBHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011133182-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2011-10-27 WO disclosed