SCHEMBL25666151

SCHEMBL25666151

COc1ccc(Nc2c(N3CCOCC3)cnc3ccc(F)cc23)c(C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.46
KCNH2 Q12809 1/20 0.45
CCNC P24863 1/20 0.45
CDK8 P49336 1/20 0.45
CSF1R P07333 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25666149 0.91 CSF1R (0.44) KCNH2CSF1R
SCHEMBL25666208 0.90 CCNC (0.45) PDE4BKCNH2CCNCCDK8CSF1R
SCHEMBL25666212 0.90 MAPT (0.50) PDE4BCSF1R
SCHEMBL25666144 0.90 RXFP1 (0.46) PDE4BKCNH2
SCHEMBL25666147 0.89 KCNH2 (0.52) KCNH2CSF1R
SCHEMBL25666146 0.87 KMT2A (0.46) KCNH2CSF1R
SCHEMBL25666124 0.85 RXFP1 (0.43) KCNH2CSF1R
SCHEMBL25666211 0.85 KMT2A (0.48) KCNH2CSF1R
SCHEMBL25665052 0.83 CNR2 (0.42) PDE4BCSF1R
SCHEMBL25665661 0.81 PDE4B (0.46) PDE4BCCNCCDK8CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023086220-A2 PAPD5 INHIBITORS AND METHODS OF USE THEREOF THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2023-05-19 WO disclosed