SCHEMBL25685294

SCHEMBL25685294

Cc1ccc(N2CC3(CCN(Cc4ccccc4)C3)CC2=O)cc1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.58
TMEM97 Q5BJF2 1/20 0.58
OPRM1 P35372 1/20 0.50
SSTR5 P35346 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25669204 0.87 SIGMAR1 (0.47) SIGMAR1TMEM97OPRM1SSTR5CYP3A4
SCHEMBL24993856 0.82 SIGMAR1 (0.54) SIGMAR1OPRM1SSTR5CYP2D6TSHR
SCHEMBL19693299 0.75 CYP2D6 (0.54) CYP3A4CYP2D6TSHR
SCHEMBL10111366 0.74 SSTR5 (0.61) SIGMAR1TMEM97SSTR5
SCHEMBL5243003 0.74 CYP2D6 (0.67) SIGMAR1CYP3A4CYP2D6TSHR
SCHEMBL25669421 0.73 TMEM97 (0.50) SIGMAR1TMEM97POLB
SCHEMBL24994297 0.73 CYP2D6 (0.55) SIGMAR1OPRM1CYP3A4CYP2D6TSHR
SCHEMBL1732446 0.73 CYP2D6 (0.65) SIGMAR1CYP3A4CYP2D6TSHR
SCHEMBL9851544 0.72 CYP2D6 (0.69) CYP3A4CYP2D6TSHRLMNA
SCHEMBL10111365 0.72 SSTR5 (0.61) SIGMAR1TMEM97OPRM1SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109883-A1 AROMATIC HETEROCYCLE-SUBSTITUTED COMPOUNDS, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2023-06-22 WO disclosed