SCHEMBL2569906

SCHEMBL2569906

O=C(O)N1CCc2nc3ccnn3c(N3CCC3CO)c2CC1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 18/20 0.44
HTR2B P41595 17/20 0.42
HTR2A P28223 16/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574733 0.88 HTR2C (0.43) HTR2CHTR2BHTR2A
SCHEMBL2574735 0.88 HTR2C (0.43) HTR2CHTR2BHTR2A
SCHEMBL9947809 0.86 HTR2C (0.41) HTR2CHTR2BHTR2A
SCHEMBL9947811 0.86 HTR2C (0.41) HTR2CHTR2BHTR2A
SCHEMBL10217195 0.83 HTR2C (0.62) HTR2CHTR2BHTR2A
SCHEMBL2573429 0.82 HTR2C (0.50) HTR2CHTR2BHTR2A
SCHEMBL9947881 0.77 HTR2C (0.40) HTR2CHTR2BHTR2A
SCHEMBL9947882 0.77 HTR2C (0.40) HTR2CHTR2BHTR2A
SCHEMBL2569024 0.76 HTR2C (0.45) HTR2CHTR2BHTR2A
SCHEMBL2565601 0.75 HTR2C (0.44) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2384328-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR PREPARING THEM Boehringer Ingelheim International GmbH (DE) 2011-11-09 EP disclosed
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed