SCHEMBL2570735

SCHEMBL2570735

CN1CCN(Cc2cc3nc(Cl)nc(C4CNCCO4)c3s2)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.40
KCNH2 Q12809 5/20 0.36
HRH1 P35367 3/20 0.36
CYP2D6 P10635 2/20 0.36
CYP3A4 P08684 1/20 0.34
PIK3R1 P27986 2/20 0.34
MTOR P42345 3/20 0.34
USP7 Q93009 2/20 0.33
MCHR1 Q99705 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28597590 0.82 KCNH2 (0.36) KCNH2HRH1CYP2D6
SCHEMBL28591605 0.81 KCNH2 (0.36) PIK3CAKCNH2HRH1CYP2D6PIK3R1
SCHEMBL28972959 0.77 KCNH2 (0.36) KCNH2HRH1CYP2D6
SCHEMBL4893967 0.72 PIK3CA (0.37) PIK3CAKCNH2HRH1CYP3A4MTOR
SCHEMBL190232 0.72 PIK3CA (0.63) PIK3CAPIK3R1MTOR
SCHEMBL16163192 0.70 PIK3CA (0.53) PIK3CAKCNH2PIK3R1MTOR
SCHEMBL17822128 0.69 ALDH1A1 (0.36) KCNH2HRH1CYP2D6CYP3A4USP7
SCHEMBL17366063 0.69 PIK3CA (0.39) PIK3CAKCNH2PIK3R1MTORMCHR1
SCHEMBL56619 0.69 PIK3CA (0.60) PIK3CAPIK3R1MTOR
SCHEMBL2575641 0.69 PIK3CA (0.43) PIK3CAKCNH2HRH1CYP2D6PIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041139-B1 PHARMACEUTICAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-11-09 EP disclosed