SCHEMBL257157

SCHEMBL257157

NC(=O)c1cc(CN2CCOCC2)c(Br)cc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.47
MAPT P10636 5/20 0.46
ALDH1A1 P00352 4/20 0.46
ABCB1 P08183 1/20 0.46
EGFR P00533 2/20 0.46
SYK P43405 1/20 0.45
KDM4E B2RXH2 4/20 0.45
HTT P42858 3/20 0.45
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
TP53 P04637 1/20 0.45
MPI P34949 1/20 0.45
SNCA P37840 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP2A13 Q16696 1/20 0.44
MAPK1 P28482 1/20 0.43
POLB P06746 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166412 0.93 CCR5 (0.50) CCR5MAPTALDH1A1ABCB1EGFR
SCHEMBL15204994 0.89 CCR5 (0.47) CCR5MAPTALDH1A1ABCB1EGFR
SCHEMBL166183 0.88 CCR5 (0.50) CCR5MAPTALDH1A1ABCB1EGFR
SCHEMBL166797 0.84 CCR5 (0.47) CCR5MAPTALDH1A1ABCB1EGFR
SCHEMBL15204854 0.80 LRRK2 (0.61) POLB
SCHEMBL167781 0.79 CCR5 (0.50) CCR5MAPTALDH1A1KDM4EHTT
SCHEMBL168123 0.77 LRRK2 (0.60) CCR5MAPTKDM4EHTTSMN1; SMN2
SCHEMBL168887 0.76 LRRK2 (0.61) POLB
SCHEMBL165453 0.76 LRRK2 (0.67)
SCHEMBL167180 0.76 PTGER1 (0.45) CCR5MAPTALDH1A1EGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028629-A1 2 - (BENZYLOXY) BENZAMIDES AS LRRK2 KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed