SCHEMBL25720199

SCHEMBL25720199

CCOc1cccc(C(=O)Cc2ccncc2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.62
HTT P42858 1/20 0.62
ROCK2 O75116 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
ROCK1 Q13464 1/20 0.52
KMT2A Q03164 3/20 0.50
HPGD P15428 3/20 0.50
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
RECQL P46063 1/20 0.50
HSD17B10 Q99714 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2477853 0.86 LMNA (0.54) LMNAHTTROCK2CYP3A4CYP2D6
SCHEMBL17088193 0.82 KMT2A (0.67) LMNAHTTKMT2AALDH1A1MAPT
SCHEMBL25720255 0.82 HPGD (0.49) LMNAHTTKMT2AHPGDALDH1A1
SCHEMBL6282499 0.80 GRM1 (0.46) LMNACYP3A4CYP2D6CYP2C9HPGD
SCHEMBL25196861 0.79 SMPD1 (0.62) RAB9ACYP19A1
SCHEMBL30391457 0.79 SMPD1 (0.62) RAB9ACYP19A1
SCHEMBL11044058 0.79 HPGD (0.56) LMNAHTTKMT2AHPGDALDH1A1
SCHEMBL3073424 0.78 NT5E (0.55) LMNAKMT2AHPGDALDH1A1MAPT
SCHEMBL1845879 0.78 MAPT (0.49) LMNACYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7913254 0.77 HPGD (0.55) LMNAHTTKMT2AHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091873-A1 GRAM-NEGATIVE SPECIFIC ANTIBIOTICS SPARING EFFECT ON GUT MICROBIOME THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-05-25 WO disclosed