SCHEMBL25746321

SCHEMBL25746321

Cn1ncc2c(S)nc(C3CC3)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.46
CHRM3 P20309 3/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HRH1 P35367 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
PDE8B O95263 1/20 0.34
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
HTR2C P28335 3/20 0.34
BCDIN3D Q7Z5W3 1/20 0.34
PDE10A Q9Y233 2/20 0.33
SHMT2 P34897 1/20 0.33
NSD2 O96028 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31391497 1.00 PDE2A (0.46) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL30095656 0.83 PDE10A (0.47) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL29174941 0.83 PDE10A (0.47) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL30095840 0.82 PDE2A (0.46) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL29174903 0.82 PDE2A (0.46) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL4698941 0.77 PDE2A (0.42) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL31391465 0.73 PDE2A (0.42) PDE2AMEN1KMT2AHRH1HRH4
SCHEMBL25746365 0.73 PDE2A (0.42) PDE2AMEN1KMT2AHRH1HRH4
SCHEMBL31391385 0.72 PDE2A (0.38) PDE2ACHRM3PDE4APDE4BPDE4C
SCHEMBL31391527 0.68 PDE2A (0.38) PDE2AMEN1KMT2AHRH1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023118507-A2 COMPOUNDS AND USE THEREOF AS HDAC6 INHIBITORS AUGUSTINE THERAPEUTICS (BE) 2023-06-29 WO disclosed