SCHEMBL2574993

SCHEMBL2574993

O=c1[nH]c2ccccc2c2c(-c3ccc4c(c3)CNCC4)csc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 1/20 0.52
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
CD274 Q9NZQ7 2/20 0.38
PNMT P11086 4/20 0.36
ASIC3 Q9UHC3 1/20 0.36
SYK P43405 2/20 0.35
CD44 P16070 1/20 0.35
MAOB P27338 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HTR5A P47898 1/20 0.34
NISCH Q9Y2I1 1/20 0.34
NR2E1 Q9Y466 1/20 0.34
CYP1A2 P05177 1/20 0.34
PPARG P37231 1/20 0.34
HTT P42858 1/20 0.34
NCOA2 Q15596 1/20 0.34
NCOA1 Q15788 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14672729 0.87 NEK1 (0.57) NEK1
Hydrochloric Acid SCHEMBL2571837 0.75 TNKS (0.50) TNKSTNKS2KDM4ECYP1A2PPARG
SCHEMBL2544993 0.74 TNKS (0.47) TNKSTNKS2KDM4ECYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL15092541 0.73 TNKS (0.46) TNKSTNKS2KDM4ECYP1A2SMN1; SMN2
SCHEMBL25404459 0.69 CD274 (0.51) CD274PNMTASIC3SYKCD44
SCHEMBL31083759 0.69 CD274 (0.51) CD274PNMTASIC3SYKCD44
SCHEMBL12279603 0.69 NEK1 (1.00) NEK1
Hydrochloric Acid SCHEMBL15092099 0.68 NEK1 (0.98) NEK1
Hydrochloric Acid SCHEMBL15092417 0.66 NEK1 (0.73) NEK1
SCHEMBL25401778 0.66 CD274 (0.52) CD274PNMTASIC3CD44MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed