SCHEMBL25401778

SCHEMBL25401778

c1ccc2c(-c3ccc4c(c3)CCNC4)c[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 3/20 0.52
HSD17B10 Q99714 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
DRD2 P14416 1/20 0.49
ALOX15 P16050 1/20 0.49
HTR2C P28335 1/20 0.49
TDO2 P48775 9/20 0.48
ASIC3 Q9UHC3 2/20 0.48
NR4A2 P43354 1/20 0.48
PNMT P11086 1/20 0.45
CD44 P16070 1/20 0.45
MAOB P27338 1/20 0.45
IMPDH2 P12268 1/20 0.44
MAPK1 P28482 1/20 0.44
ASH1L Q9NR48 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31070511 0.88 NR4A2 (0.53) HSD17B10TDO2NR4A2IMPDH2MAPK1
SCHEMBL25402840 0.77 CD274 (0.61) CD274DRD2ASIC3PNMTCD44
SCHEMBL30593259 0.74 CD274 (0.51) CD274DRD2ASIC3PNMTCD44
SCHEMBL25404671 0.74 CD274 (0.51) CD274DRD2ASIC3PNMTCD44
SCHEMBL25404459 0.74 CD274 (0.51) CD274DRD2ASIC3PNMTCD44
SCHEMBL31083759 0.74 CD274 (0.51) CD274DRD2ASIC3PNMTCD44
SCHEMBL6347388 0.74 ASIC3 (0.65) CD274DRD2ASIC3PNMTCD44
SCHEMBL4553211 0.74 CD274 (0.60) CD274DRD2ASIC3PNMTCD44
SCHEMBL28377762 0.73 NR4A2 (0.81) HSD17B10ALDH1A1MAPTTDO2NR4A2
SCHEMBL12156777 0.72 ALDH1A1 (0.47) HSD17B10KDM4EALDH1A1MAPTDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
WO-2023174383-A1 DIHYDROISOQUINOLINE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-09-21 WO disclosed