SCHEMBL25751343

SCHEMBL25751343

COC(=O)c1cc(-n2c(C)cc(OCc3ncc(C)cc3F)cc2=O)c(C)cn1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPKAPK5 Q8IW41 16/20 0.42
MAPK14 Q16539 15/20 0.42
MAPK1 P28482 14/20 0.42
MAPKAPK2 P49137 1/20 0.39
ALOX5AP P20292 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24461582 0.94 MAPKAPK5 (0.45) MAPKAPK5MAPK14MAPK1MAPKAPK2
SCHEMBL29617132 0.94 MAPKAPK5 (0.45) MAPKAPK5MAPK14MAPK1MAPKAPK2
SCHEMBL25751364 0.90 MAPKAPK5 (0.43) MAPKAPK5MAPK14MAPK1MAPKAPK2ALOX5AP
SCHEMBL25751371 0.90 MAPKAPK5 (0.43) MAPKAPK5MAPK14MAPK1MAPKAPK2ALOX5AP
SCHEMBL25751368 0.87 MAPKAPK5 (0.40) MAPKAPK5MAPK14MAPK1MAPKAPK2ALOX5AP
SCHEMBL26325986 0.85 MAPKAPK5 (0.41) MAPKAPK5MAPK14MAPK1MAPKAPK2ALOX5AP
SCHEMBL24461392 0.84 MAPKAPK5 (0.45) MAPKAPK5MAPK14MAPK1MAPKAPK2
SCHEMBL29617129 0.84 MAPKAPK5 (0.45) MAPKAPK5MAPK14MAPK1MAPKAPK2
SCHEMBL24461685 0.84 MAPKAPK5 (0.47) MAPKAPK5MAPK14MAPK1MAPKAPK2
SCHEMBL29617114 0.84 MAPKAPK5 (0.45) MAPKAPK5MAPK14MAPK1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS, INC. 2023-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS PIR, PUM1, ZRANB2 MAPKAPK5 848/4885MAPK14 2275/4885MAPK1 924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.