SCHEMBL25751761

SCHEMBL25751761

CNC(=O)c1cc(-n2c(C)cc(OCc3ccc(F)cc3F)c(Cl)c2=O)c(C)cn1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 18/20 0.61
ROCK2 O75116 1/20 0.61
MAPK12 P53778 1/20 0.61
MAPK11 Q15759 1/20 0.61
STRADA Q7RTN6 1/20 0.61
MAPKAPK2 P49137 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9111868 0.90 MAPKAPK2 (0.62) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL9110526 0.90 MAPKAPK2 (0.64) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL9109111 0.90 MAPKAPK2 (0.66) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL24461663 0.88 MAPKAPK5 (0.59) MAPK14MAPKAPK2
SCHEMBL4377493 0.86 MAPK14 (0.82) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL24461461 0.85 MAPKAPK2 (0.59) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4376468 0.84 MAPK14 (0.82) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4378073 0.83 MAPK14 (0.82) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL29593154 0.83 MAPK14 (0.82) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4488757 0.82 MAPK14 (0.85) MAPK14ROCK2MAPK12MAPK11STRADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11767309-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds ACLARIS THERAPEUTICS, INC. (US) 2023-09-26 US disclosed
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS, INC. 2023-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11767309-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds PIR, PUM1, ZRANB2 MAPK14 2275/4885ROCK2 2348/4885MAPK12 1518/4885
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS PIR, PUM1, ZRANB2 MAPK14 2275/4885ROCK2 2348/4885MAPK12 1518/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.