SCHEMBL25755670

SCHEMBL25755670

N#Cc1c[nH]c(=O)c2c(Br)csc12

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPYD Q12882 1/20 0.41
MCL1 Q07820 10/20 0.40
CHEK1 O14757 2/20 0.38
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
DYRK1A Q13627 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CHUK O15111 2/20 0.33
CDK2 P24941 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27174968 0.75 DYRK1A (0.47) DPYDMCL1DYRK1ACHUK
SCHEMBL3528687 0.74 PDPK1 (0.39) ALDH1A1GSK3B
SCHEMBL4474629 0.74 DPYD (0.35) DPYDALDH1A1GSK3B
SCHEMBL25754505 0.74 GPR35 (0.33) ALDH1A1GSK3B
SCHEMBL31128869 0.70 KDM4E (0.42) CHEK1DYRK1AKDM4EGSK3B
SCHEMBL3088202 0.69 GSK3B (0.41) DPYDMCL1CHEK1PIK3CDPIK3CA
SCHEMBL3069636 0.68 DPYD (0.42) DPYDMCL1PIK3CDPIK3CAPIK3CB
SCHEMBL25755671 0.68 KDM4E (0.38) KDM4EALDH1A1
SCHEMBL3617645 0.66 TNKS (0.47) DPYDMCL1DYRK1AKDM4EALDH1A1
SCHEMBL3086572 0.66 DPYD (0.40) DPYDMCL1CHEK1PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024208315-A1 AROMATIC HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 中国医药研究开发中心有限公司 2024-10-10 WO disclosed
WO-2023109954-A1 TYK2 INHIBITORS AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO. LTD. (CN) 2023-06-22 WO disclosed