SCHEMBL257587

SCHEMBL257587

COc1cc2ncc3c(c2cc1CCc1cccs1)n(-c1c(F)cc(C#N)cc1F)c(=O)n3C

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 9/20 0.63
ATM Q13315 4/20 0.50
GRM4 Q14833 2/20 0.37
MAP2K1 Q02750 1/20 0.36
PIK3CD O00329 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
MTOR P42345 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
KCNH2 Q12809 2/20 0.35
AKT1 P31749 1/20 0.34
KIT P10721 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15064201 0.89 PRKDC (0.60) PRKDCATMMAP2K1KIT
SCHEMBL10059179 0.88 PRKDC (0.68) PRKDCATMGRM4MAP2K1PIK3CD
SCHEMBL256582 0.81 PRKDC (0.74) PRKDCATMPIK3CDPIK3CAPIK3CB
SCHEMBL15064831 0.80 PRKDC (0.58) PRKDCATMGRM4
SCHEMBL10059983 0.80 PRKDC (0.57) PRKDCATMGRM4PIK3CDPIK3CA
SCHEMBL15064295 0.80 PRKDC (0.73) PRKDCATMMAP2K1KIT
SCHEMBL15064494 0.80 PRKDC (0.59) PRKDCATMGRM4PIK3CDPIK3CA
SCHEMBL10059173 0.79 PRKDC (0.82) PRKDCATMGRM4MAP2K1PIK3CD
SCHEMBL257190 0.78 PRKDC (0.66) PRKDCATMMAP2K1KIT
SCHEMBL167275 0.78 PRKDC (1.00) PRKDCATMMAP2K1PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028233-A1 IMIDAZO[4,5-C]QUINOLINES AS DNA-PK INHIBITORS MERCK PATENT GMBH (DE) 2012-03-08 WO disclosed