SCHEMBL25773255

SCHEMBL25773255

COc1cc2c(cc1OC)-c1c/c(=N\c3c(C)cc(C(F)(F)F)cc3C)[nH]c(=O)n1CC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 8/20 0.54
MAPK1 P28482 8/20 0.54
MAPT P10636 4/20 0.54
CYP3A4 P08684 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
PDE4A P27815 2/20 0.54
PDE4B Q07343 2/20 0.54
PDE4C Q08493 2/20 0.54
PDE4D Q08499 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
ABCC4 O15439 1/20 0.54
ABCC5 O15440 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
NFKB1 P19838 1/20 0.54
CYP2C19 P33261 1/20 0.54
THPO P40225 1/20 0.54
HIF1A Q16665 1/20 0.54
KMT2A Q03164 5/20 0.53
LMNA P02545 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25773363 0.90 TSHR (0.56) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL11967263 0.90 TSHR (0.66) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL31619806 0.90 TSHR (0.66) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL5113232 0.90 TSHR (0.66) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL5113231 0.90 TSHR (0.66) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL31632614 0.86 TSHR (0.59) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL31620968 0.86 TSHR (0.59) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL25773302 0.85 MAPK1 (0.53) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL31620981 0.84 TSHR (0.56) TSHRMAPK1MAPTCYP3A4TDP1
SCHEMBL31620970 0.84 TSHR (0.53) TSHRMAPK1MAPTCYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109802-A1 TRICYCLIC FUSED HETEROCYCLIC PDE3/4 DUAL INHIBITOR AND USE THEREOF 海思科医药集团股份有限公司 2023-06-22 WO disclosed